The AAPS journalAprepitantBiological AvailabilityFreeze DryingNanoparticlesAdministration
A Novel Oral Disintegrating Tablet Containing Aprepitant Nanocrystal Developed by Freeze-Drying Technology: An Effective Strategy to Enhance Aprepitant Bioavailability.
Yutong Li, Meihui Yi, Keke Ma, Jingxin Gou, Tian Yin, Yu Zhang, Xing Tang, Haibing He
Published: 202510.1208/s12248-025-01187-7
Abstract
This study developed a novel aprepitant (APT) nanocrystal-containing oral disintegrating tablet (ODT) to enhance the oral bioavailability of APT through "rapid disintegration". APT nanocrystal suspension (APT-NS) was prepared via miniaturized media m…
Preview only. Read the full abstract at the source