Nature chemical biology
Complex-specific inhibitors for interrogating ATAC histone acetyltransferase complex.
Sha Liu, Jinzhao Liu, Yinqiao Wu, Xinyi Yao, Xiang Li, Xinyu Dong, Qi Li, Hayden Jit Hei Cheung, Kwan Yuen Wong, Yuanyuan Li, Mu He, Chi-Leung Chiang, Jason Wing Hon Wong, Haitao Li, Weiping Wang
Published: 202610.1038/s41589-025-02132-7
Abstract
Histone acetyltransferases (HATs) modify chromatin to regulate gene expression. Instead of acting alone, HATs function in complexes with other proteins, leading to variations in substrate specificity, genomic localization and cellular function. To un…
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