Journal of medicinal chemistryDrug DiscoveryKineticsHumansChemistryPharmaceutical
Innovative Medicinal Chemistry Strategies for Improving Target Binding Kinetics in Drug Discovery.
Hui Qiao, Ziqiao Yuan, Lulu Xing, Bao-Xia He, Li-Ying Ma, Zhang-Xu He
Published: 202510.1021/acs.jmedchem.5c02299
Abstract
The concept of drug-target binding kinetics has garnered significant attention in recent drug discovery literature. Incorporating drug-target binding kinetics into the early phases of drug development has resulted in several clinical candidates exhib…
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