Journal of medicinal chemistryAnimalsHumansPhenforminPancreatic NeoplasmsMitochondria
Re/99mTc Tricarbonyl Phenformin Complexes Targeting Mitochondria as Pancreatic Cancer Theranostics.
Chiyi Xiong, Boping Jing, Qizhen Cao, Junjie Li, Merve Alpay, Haiyan Chen, Wai-Kin Chan, Huamin Wang, Amir M Gholizadeh, Diana S-L Chow, Chun Li
Published: 202510.1021/acs.jmedchem.5c01760
Abstract
Phenformin has antitumor effects against pancreatic cancer. We report a phenformin complex with the technetium-99m tricarbonyl [99mTc(CO)3], termed 99mTc-Phen, that permitted noninvasive visualization of tumor uptake in models of pancreatic cancer by…
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