Biochemical pharmacologyHumansQuinolinesAllosteric RegulationQuinoxalinesReceptor
Discovery and characterization of quinoxaline and quinoline carboxamides as allosteric cannabinoid receptor modulators.
Chunyang Bi, Andhika B Mahardhika, Thanigaimalai Pillaiyar, Christa E Müller
Published: 202610.1016/j.bcp.2025.117485
Abstract
Cannabinoid (CB) receptors type 1 (CB1) and type 2 (CB2) are Gi protein-coupled receptors that play important roles in brain function and immune regulation. While orthosteric CB1 and CB2 receptor agonists and antagonists have been widely studied, onl…
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