Archiv der PharmazieCarbonic Anhydrase InhibitorsStructure-Activity RelationshipTetrazolesEscherichia coliCarbonic Anhydrases
Tetrazole Derivatives as Multiclass Inhibitors of Bacterial Carbonic Anhydrases.
Andrea Ammara, Simone Giovannuzzi, Viviana De Luca, Clemente Capasso, Alessio Nocentini, Claudiu T Supuran, Paola Gratteri
Published: 202510.1002/ardp.70177
Abstract
This study investigates derivatives including a tetrazole zinc-binding group as inhibitors of the α-, β-, and γ-class carbonic anhydrase (CA) isoforms from pathogenic bacteria such as Vibrio cholerae, Escherichia coli, and Streptococcus mutans. A lib…
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