Angewandte Chemie (International ed. in English)Mycobacterium tuberculosisPyrazinesAntitubercular AgentsMicrobial Sensitivity TestsHumans
Discovery and Total Synthesis of Crossiguanipyrazines with Potent Activity Against Mycobacterium tuberculosis.
Haowen Zhao, Etienne Bickel, Jiaqi Liu, Xiaoli Yang, Michael Dal Molin, Jason Chhen, Shuqin Liu, Haiyan Sui, Xiaoying Bian, Xiaoyi Wei, Jan Rybniker, Uli Kazmaier, Chengzhang Fu
Published: 202510.1002/anie.202513977
Abstract
Tuberculosis (TB), caused by Mycobacterium tuberculosis, remains one of the most devastating infectious diseases, with rising antimicrobial resistance exacerbating the urgent need for new therapeutic agents. Here, we report the discovery of crossigua…
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